产品详情
产品名称SB366791
简述Inhibitors
纯化98.00%
生物活性SB-366791 is a novel, potent, and selective, cinnamide TRPV1 antagonist.
基因/蛋白名称TRP/TRPV Channel inhibitor
CAS号472981-92-3
计算分子量287.74
配方C16H14ClNO2
保存3 years -20˚C powder;2 years -80˚C in solvent;
产品描述
Research Area:Others
SMILES:COC1=CC=CC(=C1)NC(=O)/C=C/C2=CC=C(C=C2)Cl
Pathways:Membrane transporter/Ion channel
Receptor:TRPV1
Boling pt:
Melting pt:
Solubility:Ethanol: <1 mg/mLDMSO: 57 mg/mL (198.09 mM)
Water: <1 mg/mL
Appearance:
Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.
背景文献
1. Gunthorpe MJ,et al. Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist. Neuropharmacology. 2004 Jan;46(1):133-49.
The lead time is currently 7-30 days.
